PHARMACOPEIA, INC.

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Technologies

Intl Class Technology # of Patents Rank
 
 
 
C07D HETEROCYCLIC COMPOUNDS 16106
 
 
 
A61K PREPARATIONS FOR MEDICAL, DENTAL, OR TOILET PURPOSES 14180
 
 
 
A61P THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS 438
 
 
 
A01N PRESERVATION OF BODIES OF HUMANS OR ANIMALS OR PLANTS OR PARTS THEREOF 369
 
 
 
C25B ELECTROLYTIC OR ELECTROPHORETIC PROCESSES FOR THE PRODUCTION OF COMPOUNDS OR NON- METALS; APPARATUS THEREFOR 120

Top Patents (by citation)

Patent # Title Filing Date Issue Date Intl Class Cited #
5,798,035 High throughput solid phase chemical synthesis utilizing thin cylindrical reaction vessels useable for biological assayOct 03, 96Aug 25, 98[C25B]37
7,417,045 Heterocyclic substituted pyridine or phenyl compounds with CXCR3 antagonist activityFeb 14, 06Aug 26, 08[A61K]18
6,903,131 3,4-di-substituted maleimide compounds as CXC chemokine receptor antagonistsOct 11, 02Jun 07, 05[C07D, A61K]8
7,253,174 N-heterocyclic inhibitors of TNF-.alpha. expressionJul 12, 06Aug 07, 07[C07D]5
7,786,124 Heterocyclic substituted pyridine compounds with CXCR3 antagonist activityMar 19, 07Aug 31, 10[C07D, A61K]2
7,700,592 α2C adrenoreceptor agonistsFeb 13, 07Apr 20, 10[C07D, A61K]2
7,479,495 N-heterocyclic inhibitors of TNF-α expressionJun 02, 05Jan 20, 09[C07D, A61P, A61K]2
7,763,609 Heterocyclic aspartyl protease inhibitorsFeb 23, 07Jul 27, 10[C07D, A61K]1
7,763,616 Piperazine-piperidines with CXCR3 antagonist activityFeb 14, 06Jul 27, 10[C07D, A61P, A61K]1
6,943,161 Pyrimidine and triazine kinase inhibitorsJun 28, 02Sep 13, 05[C07D, A61P, A61K]1

Recent Publications

Publication # Title Filing Date Pub Date Intl Class
2012/0276,118 HETEROCYCLIC ASPARTYL PROTEASE INHIBITORSMar 14, 12Nov 01, 12[A61K]
2012/0231,017 HETEROCYCLIC ASPARTYL PROTEASE INHIBITORSMar 08, 12Sep 13, 12[C07F, C07D, A61P, A61K]
2012/0231,018 HETEROCYCLIC ASPARTYL PROTEASE INHIBITORSMar 09, 12Sep 13, 12[A61P, A61K]
2010/0292,203 HETEROCYCLIC ASPARTYL PROTEASE INHIBITORSJan 26, 10Nov 18, 10[C07D, A61K]
2010/0197,562 FUNCTIONALLY SELECTIVE ALPHA2C ADRENORECEPTOR AGONISTSFeb 11, 08Aug 05, 10[C07D, A61P, A61K]
2009/0306,079 3,4-DI-SUBSTITUTED CYCLOBUTENE-1,2-DIONES AS CXC-CHEMOKINE RECEPTOR LIGANDSJan 13, 09Dec 10, 09[C07D, A61P, A61K]
2009/0264,416 N-BENZYL,N'-ARYLCARBONYLPIPERAZINE DERIVATIVESAug 19, 08Oct 22, 09[C07D, A61K]
2009/0005,568 Substituted 2-aminothiazoles for treating neurodegenerative diseasesAug 18, 06Jan 01, 09[C07D, A61P, A61K]
2008/0292,589 NOVEL HETEROCYCLIC SUBSTITUTED PYRIDINE OR PHENYL COMPOUNDS WITH CXCR3 ANTAGONIST ACTIVITYJun 26, 08Nov 27, 08[C07D, A61P, A61K]
2008/0214,553 2-(4-Oxo-4H-Quinazolin-3-Yl) Acetamides and Their Use as Vasopressin V3 AntagonistsMar 10, 06Sep 04, 08[C07D, A61K]

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Recent Patents

Patent # Title Filing Date Issue Date Intl Class
8,314,091 N-benzyl,N'-arylcarbonylpiperazine derivativesAug 19, 08Nov 20, 12[A01N, C07D, A61K]
8,183,252 Heterocyclic aspartyl protease inhibitorsJan 26, 10May 22, 12[A01N, C07D, A61K]
8,044,040 N-heterocyclic inhibitors of TNF-alpha expressionJul 16, 07Oct 25, 11[C07D, A61K]
8,017,616 Heterocyclic substituted pyridine compounds with CXCR3 antagonist activityDec 21, 09Sep 13, 11[C07D, A61K]
8,003,624 Functionally selective ALPHA2C adrenoreceptor agonistsFeb 13, 07Aug 23, 11[A01N, C07D]
7,951,803 8-heteroarylpurine MNK2 inhibitors for treating metabolic disordersMar 09, 07May 31, 11[C07D, A61P, A61K]
7,906,504 -isoquinolin-2-yl)acetamide derivativesSep 10, 07Mar 15, 11[C07D, A61K]
7,902,199 Heterocyclic substituted piperazine compounds with CXCR3 antagonist activityJul 12, 07Mar 08, 11[C07D, A61K]
7,820,649 Quinazolinone and isoquinolinone acetamide derivativesSep 10, 07Oct 26, 10[C07D]
7,807,686 2-(4-oxo-4H-quinazolin-3-yl)acetamides and their use as vasopressin V3 antagonistsMar 10, 06Oct 05, 10[A61K]

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Top Inventors for This Owner

Inventor Name Address # of Patent/Pub
Baldwin John J
Gwynedd Valley, PA
11
Hobbs Douglas W
Yardley, PA
10
Lai Gaifa
Edison, NJ
9
McGuinness Brian F
Plainsboro, NJ
9
Rosenblum Stuart B
West Orange, NJ
9
Dolle III Roland Ellwood
King of Prussia, PA
8
Guo Tao
Dayton, NJ
8
Henderson Ian
Hopewell, NJ
8
Li Ge
Shanghai, CN
8
Ohlmeyer Michael
Plainsboro, NJ
8