THERAVANCE BIOPHARMA R&D IP, LLC

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Patent Activity in the Last 10 Years

Technologies

Intl Class Technology Matters Rank in Class
 
 
 
A61K PREPARATIONS FOR MEDICAL, DENTAL, OR TOILET PURPOSES 27559
 
 
 
C07D HETEROCYCLIC COMPOUNDS 24126
 
 
 
C07C ACYCLIC OR CARBOCYCLIC COMPOUNDS 6475
 
 
 
A01N PRESERVATION OF BODIES OF HUMANS OR ANIMALS OR PLANTS OR PARTS THEREOF 4551
 
 
 
A61P THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS 940
 
 
 
C07F ACYCLIC, CARBOCYCLIC, OR HETEROCYCLIC COMPOUNDS CONTAINING ELEMENTS OTHER THAN CARBON, HYDROGEN, HALOGEN, OXYGEN, NITROGEN, SULFUR, SELENIUM, OR TELLURIUM 664
 
 
 
G01N INVESTIGATING OR ANALYSING MATERIALS BY DETERMINING THEIR CHEMICAL OR PHYSICAL PROPERTIES 4202
 
 
 
C12Q MEASURING OR TESTING PROCESSES INVOLVING ENZYMES OR MICRO-ORGANISMS 3122
 
 
 
A61M DEVICES FOR INTRODUCING MEDIA INTO, OR ONTO, THE BODY 2152
 
 
 
C07H SUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS 198

Top Patents (by citation)

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Recent Publications

Publication # Title Filing Date Pub Date Intl Class
2018/0051,023 NEPRILYSIN INHIBITORSJun 30, 17Feb 22, 18[A61K, C07D, C07C]

Recent Patents

Patent # Title Filing Date Issue Date Intl Class
9884807 Neprilysin inhibitorsApr 28, 17Feb 06, 18[A61K, C07F, C07D, C07C]
9872855 (2R,4R)-5-(5′-Chloro-2′-fluorobiphenyl-4-yl)-2-hydroxy-4-[(5-methyloxazole-2-carbonyl)amino]pentanoic acidNov 21, 16Jan 23, 18[A61K, C07D]
9873685 Neprilysin inhibitorsApr 26, 17Jan 23, 18[A61K, C07D]
9873692 Quinolinone-carboxamide compounds as 5-HT4 receptor agonistsMar 15, 17Jan 23, 18[C07D]
9873696 Neprilysin inhibitorsDec 14, 16Jan 23, 18[A61K, C07D]
9868698 (2S,4R)-5-(5′-chloro-2′-fluorobiphenyl-4-yl)-4-(ethoxyoxalylamino)-2-hydroxymethyl-2-methylpentanoic acidApr 28, 17Jan 16, 18[C07C]
9845332 Neprilysin inhibitorsMay 19, 17Dec 19, 17[A61K, C07D]
9839639 Neprilysin inhibitorsJan 19, 17Dec 12, 17[A61K, C07D, C07C]
9840460 Neprilysin inhibitorsMay 22, 17Dec 12, 17[A61K, C07D, C07C]
9828367 Neprilysin inhibitorsJul 21, 16Nov 28, 17[A61K, C07D]

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Expired/Abandoned/Withdrawn Patents

Patent # Title Status Filing Date Issue/Pub Date Intl Class
2016/0287,573 COMBINATION DOSAGE FORM OF A MU OPIOID RECEPTOR ANTAGONIST AND AN OPIOID AGENTAbandonedMar 31, 16Oct 06, 16[A61K]
2016/0022,660 CRYSTALLINE FORM OF A 4-[2-(2-FLUOROPHENOXYMETHYL)PHENYL]PIPERIDINE COMPOUNDAbandonedJun 02, 15Jan 28, 16[A61K]
2015/0141,483 CRYSTALLINE FORMS OF A 3-[2-METHANESULFONYL-1-(4-TRIFLUOROMETHYL-PHENOXY)ETHYL]PYRROLIDINE COMPOUNDAbandonedJan 26, 15May 21, 15[A61K]
2015/0119,571 NEPRILYSIN INHIBITORSAbandonedSep 04, 14Apr 30, 15[C07F, C07D]
2015/0011,597 DUAL-ACTING ANTIHYPERTENSIVE AGENTSAbandonedMar 27, 14Jan 08, 15[C07D, C07C]
2014/0057,939 5-HT4 RECEPTOR AGONIST COMPOUNDS FOR TREATMENT OF COGNITIVE DISORDERSAbandonedFeb 20, 13Feb 27, 14[A61K]
2013/0324,550 1-(2-PHENOXYMETHYLHETEROARYL) PIPERIDINE AND PIPERAZINE COMPOUNDSAbandonedAug 09, 13Dec 05, 13[C07D]
2013/0273,568 BENZIMIDAZOLE-CARBOXAMIDE COMPOUNDS AS 5-HT4 RECEPTOR AGONISTSAbandonedJan 16, 13Oct 17, 13[G01N]
2013/0274,288 BIPHENYL COMPOUNDS USEFUL AS MUSCARINIC RECEPTOR ANTAGONISTSAbandonedJun 11, 13Oct 17, 13[C07D]
2012/0071,654 ARYL ANILINE DERIVATIVES AS BETA2 ADRENERGIC RECEPTOR AGONISTSAbandonedJun 28, 11Mar 22, 12[C07D, C07C]
2011/0263,631 COMBINATION OF A SEROTONIN AND NOREPINEPHRINE REUPTAKE INHIBITOR AND AN OPIOID AGONIST FOR THE TREATMENT OF PAINAbandonedApr 21, 11Oct 27, 11[A61K, C12Q, A61P]
2011/0257,243 3-PHENOXYMETHYLPYRROLIDINE COMPOUNDSAbandonedJun 30, 11Oct 20, 11[A61K, C07D, A61P]
7981931 Pharmaceutical compositions of short-acting sedative hypnotic agentExpiredDec 02, 09Jul 19, 11[A61K, A01N]
2010/0267,743 3-(PHENOXYPYRROLIDIN-3-YL-METHYL)HETEROARYL, 3-(PHENYLPYRROLIDIN-3-YLMETHOXY)HETEROARYL, AND 3-(HETEROARYLPYRROLIDIN-3-YLMETHOXY)HETEROARYL COMPOUNDSAbandonedApr 14, 10Oct 21, 10[A61K, C07D, A61P]
7790766 Pharmaceutical compositions of short-acting sedative hypnotic agentExpiredJul 21, 04Sep 07, 10[A61K]
2010/0137,325 BIPHENYL COMPOUNDS USEFUL AS MUSCARINIC RECEPTOR ANTAGONISTSAbandonedFeb 03, 10Jun 03, 10[A61K, C07D, A61P]
2010/0112,661 ONCOKINASE FUSION POLYPEPTIDES ASSOCIATED WITH HYPERPROLIFERATIVE AND RELATED DISORDERS, NUCLEIC ACIDS ENCODING THE SAME AND METHODS FOR DETECTING AND IDENTIFYING THE SAMEAbandonedAug 26, 09May 06, 10[C12N]
2010/0048,622 CRYSTALLINE FORMS OF A BIPHENYL COMPOUNDAbandonedSep 21, 09Feb 25, 10[A61K, A61P]
2009/0306,134 Muscarinic receptor antagonistsAbandonedSep 30, 08Dec 10, 09[A61K, C07D]
7514425 Short-acting sedative hypnotic agents for anesthesia and sedationExpiredJan 13, 06Apr 07, 09[A61K]

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