VERTEX PHARMACEUTICALS INCORPORATED

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Patent Activity in the Last 10 Years

Technologies

Intl Class Technology Matters Rank in Class
 
 
 
A61K PREPARATIONS FOR MEDICAL, DENTAL, OR TOILET PURPOSES 43633
 
 
 
C07D HETEROCYCLIC COMPOUNDS 42912
 
 
 
A01N PRESERVATION OF BODIES OF HUMANS OR ANIMALS OR PLANTS OR PARTS THEREOF 4749
 
 
 
G01N INVESTIGATING OR ANALYSING MATERIALS BY DETERMINING THEIR CHEMICAL OR PHYSICAL PROPERTIES 44162
 
 
 
A61P THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS 3516
 
 
 
C07C ACYCLIC OR CARBOCYCLIC COMPOUNDS 32106
 
 
 
C12N MICRO-ORGANISMS OR ENZYMES; COMPOSITIONS THEREOF 32135
 
 
 
C07K PEPTIDES 28108
 
 
 
C12Q MEASURING OR TESTING PROCESSES INVOLVING ENZYMES OR MICRO-ORGANISMS 22103
 
 
 
C12P FERMENTATION OR ENZYME-USING PROCESSES TO SYNTHESISE A DESIRED CHEMICAL COMPOUND OR COMPOSITION OR TO SEPARATE OPTICAL ISOMERS FROM A RACEMIC MIXTURE 1287

Top Patents (by citation)

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Recent Publications

Publication # Title Filing Date Pub Date Intl Class
2018/0008,546 FORMULATIONS OF 3-(6-(1-(2,2-DIFLUOROBENZO[D][1,3]DIOXOL-5-YL) CYCLOPROPANECARBOXAMIDO)-3-METHYLPYRIDIN-2-YL)BENZOIC ACIDJul 20, 17Jan 11, 18[A61J, A61K]
2017/0327,456 PROCESS FOR MAKING MODULATORS OF CYSTIC FIBROSIS TRANSMEMBRANE CONDUCTANCE REGULATORAug 02, 17Nov 16, 17[C07C]
2017/0204,478 INFLUENZA A VIRUS VARIANTSMar 31, 17Jul 20, 17[C12Q, C12N, G01N, G06F, C07K]
2017/0204,479 INFLUENZA A VIRUS VARIANTSMar 31, 17Jul 20, 17[C12Q, C12N, G01N, C07K]
2017/0174,675 Modulators of Cystic Fibrosis Transmembrane Conductance RegulatorApr 22, 16Jun 22, 17[C07D]
2017/0107,205 MODULATORS OF ATP-BINDING CASSETTE TRANSPORTERSJun 01, 16Apr 20, 17[C07D]
2017/0087,144 PHARMACEUTICAL COMPOSITION AND ADMINISTRATIONS THEREOFAug 31, 16Mar 30, 17[A61K]
2016/0355,512 INHIBITORS OF INFLUENZA VIRUSES REPLICATIONJun 09, 16Dec 08, 16[A61K, C07D]
2016/0324,846 Pharmaceutical Compositions for the Treatment of CFTR Mediated DiseasesMay 11, 16Nov 10, 16[A61K]
2016/0318,931 MODULATORS OF ATP-BINDING CASSETTE TRANSPORTERSFeb 29, 16Nov 03, 16[A61K, C07D, C07C, G01N]

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Recent Patents

Patent # Title Filing Date Issue Date Intl Class
9908878 Inhibitors of influenza viruses replicationJun 09, 16Mar 06, 18[A61K, C07F, C07D]
9890176 Mannose derivatives for treating bacterial infectionsMar 12, 14Feb 13, 18[C07H, C07D]
9878993 DNA-PK inhibitors for treatment of cancerMay 19, 16Jan 30, 18[C07D]
9862709 Processes for making compounds useful as inhibitors of ATR kinaseApr 03, 15Jan 09, 18[C07D, C07C]
9856248 Modulators of cystic fibrosis transmembrane conductance regulatorApr 22, 16Jan 02, 18[A61K, C07D]
9840499 Solid forms of 3-(6-(1-(2,2-difluorobenzo[d][1,3]dioxol-5-yl)cyclopropanecarboxamido)-3-methylpyridin-2-yl) benzoic acidApr 12, 16Dec 12, 17[A61K, C07D]
9828397 Prodrugs of pyridone amides useful as modulators of sodium channelsSep 09, 16Nov 28, 17[A61K, C07F]
9808459 Inhibitors of influenza viruses replicationOct 21, 16Nov 07, 17[A61K, C07D]
9791456 Method for measuring ATR inhibition mediated increases in DNA damageFeb 27, 15Oct 17, 17[G01N]
9782408 Modulators of cystic fibrosis transmembrane conductance regulatorOct 06, 15Oct 10, 17[A61J, A61K, C07D]

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Expired/Abandoned/Withdrawn Patents

Patent # Title Status Filing Date Issue/Pub Date Intl Class
2017/0107,206 MODULATORS OF ATP-BINDING CASSETTE TRANSPORTERSAbandonedJun 03, 16Apr 20, 17[C07D]
2016/0354,381 DNA-PK INHIBITORSAbandonedMay 06, 16Dec 08, 16[A61K]
2016/0326,180 COMPOUNDS USEFUL AS INHIBITORS OF ATR KINASEAbandonedMay 03, 16Nov 10, 16[A61K, C07D, A61N]
2016/0324,788 FORMULATIONS OF 3-(6-(1-(2,2-DIFLUOROBENZO[D][1,3]DIOXOL-5-YL) CYCLOPROPANECARBOXAMIDO)-3-METHYLPYRIDIN-2-YL)BENZOIC ACIDAbandonedApr 07, 16Nov 10, 16[A61K]
2016/0311,809 COMPOUNDS USEFUL AS INHIBITORS OF ATR KINASEAbandonedApr 29, 16Oct 27, 16[C07D]
2016/0271,129 COMPOUNDS USEFUL AS INHIBITORS OF ATR KINASEAbandonedMar 18, 16Sep 22, 16[A61K, C07D]
2016/0228,414 MODULATORS OF ATP-BINDING CASSETTE TRANSPORTERSAbandonedJan 29, 16Aug 11, 16[A61K]
2016/0221,952 MODULATORS OF CYSTIC FIBROSIS TRANSMEMBRANE CONDUCTANCE REGULATORAbandonedDec 31, 15Aug 04, 16[A61K, C07D, G01N]
2016/0200,684 Pharmaceutical Compositions for the Treatment of CFTR-Mediated DisordersAbandonedNov 26, 14Jul 14, 16[A61K, C07D]
2016/0166,540 MODULATORS FOR ATP-BINDING CASSETTE TRANSPORTERSAbandonedJan 11, 16Jun 16, 16[A61K, C07D]
2016/0143,898 MODULATORS OF ATP-BINDING CASSETTE TRANSPORTERSAbandonedOct 28, 15May 26, 16[A61K]
2016/0067,239 PHARMACEUTICAL COMPOSITIONS AND ADMINISTRATIONS THEREOFAbandonedJan 23, 15Mar 10, 16[A61K, G01N]
2016/0039,800 DOSAGE UNITS OF 3-(6-(1-(2,2-DIFLUOROBENZO[D] [1,3] DIOXOL-5-YL) CYCLOPROPANECARBOXAMIDO)-3-METHYLPYRIDIN-2-YL)BENZOIC ACIDAbandonedOct 22, 15Feb 11, 16[A61K, C07D]
2016/0030,406 CORRECTORS ACTING THROUGH MSD1 OF CFTR PROTEINAbandonedMar 14, 14Feb 04, 16[A61K, G01N]
2016/0022,665 Pharmaceutical Compositions and Administrations ThereofAbandonedFeb 25, 15Jan 28, 16[A61K, G01N]
2016/0022,664 Pharmaceutical Compositions and Administrations ThereofAbandonedFeb 23, 15Jan 28, 16[A61K, C12Q]
2016/0009,723 COMPOUNDS USEFUL AS INHIBITORS OF ATR KINASEAbandonedJul 15, 15Jan 14, 16[C07D]
2016/0008,359 AZAINDOLES USEFUL AS INHIBITORS OF JANUS KINASESAbandonedJul 29, 15Jan 14, 16[A61K]
2015/0376,187 COMPOUNDS USEFUL AS INHIBITORS OF ATR KINASEAbandonedJun 24, 15Dec 31, 15[A61K, C07D, A61N]
2015/0336,898 Prodrugs of Modulators of ABC TransportersAbandonedAug 04, 15Nov 26, 15[A61K, C12Q, C07F, C07D]

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