US Patent Application No: 2001/0025,041

Amidino protease inhibitors

Stats

Sep 27, 2001
Publication date
May 9, 2001
filing date
09/851,123
serial no
Granted
status

ALSO PUBLISHED AS: 6414020

Importance

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Abstract

Amidino and benzamidino compounds, including compounds of the formula: 1 wherein R.sup.1-R.sup.4, R.sup.6-R.sup.9, Y, Z, n and m are set forth in the specification, as well as hydrates, solvates or pharmaceutically acceptable salts thereof, that inhibit a number of proteolytic enzymes are described. Also described are methods for preparing the compounds of Formula I.

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First Claim

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Patent Owner(s)

Patent Owner	Address	Total Patents
3-DIMENSIONAL PHARMACEUTICALS, INC.	EXTON, PA	75

International Classification(s)

A61K:PREPARATIONS FOR MEDICAL, DENTAL, OR TOILET PURPOS....

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[Patents Count]

Inventor(s)

Inventor Name	Address	# of filed Patents	Total Citations
Illig, Carl R	-	5	1
Lu, Tianbao	-	19	11
Soll, Richard M	-	6	1
Tomczuk, Bruce E	-	10	2

Patent Citation Ranking

Forward Cites

Patent Info	(Count)	# Cites	Year
ASTRAZENECA AB (1)
7,074,820 Amidino derivatives and their use as thrombin inhibitors		0	2001

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