
US Patent No: 4,689,320
Number of patents in Portfolio can not be more than 2000
Method for inhibiting propagation of virus and anti-viral agent
Stats
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Aug 25, 1987
Issued date -
Oct 15, 1984
filing date -
06/661,204
serial no -
Expired
status

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Forward Citations
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Abstract
Described is a method for inhibiting propagation of virus which comprises delivering one or more oligodeoxynucleotides or polydeoxynucleotides to a place where a messenger RNA (mRNA) generated on propagation of the virus exists, characterized in that the oligodeoxynucleotides or polydeoxynucleotides are identical in DNA sequence with a portion of the structure of DNA hybridizable to the mRNA, the structure being capable of hybridizing to the mRNA. Also described is an anti-viral agent which comprises an effective amount of one or more oligodeoxynucleotides or polydeoxynucleotides with a conventional liquid vehicle or excipient, characterized in that the oligodeoxynucleotides or polydeoxynucleotides are identical in DNA sequence with a portion of the structure of DNA hybridizable to an mRNA generated on propagation of the virus, the structure being capable of hybridizing to the mRNA. The method and the agent can widely be applied to the treatment of viral diseases.
First Claim
Related Publications
- 15 United States
- 10 France
- 8 Japan
- 7 China
- 5 Korea
- 2 Other
Patent Owner(s)
| Patent Owner | Address | Total Patents |
|---|---|---|
| ISIS PHARMACEUTICALS, INC. | CARLSBAD, CA | 963 |
International Classification(s)
- [Classification Symbol]
- [Patents Count]
Inventor(s)
| Inventor Name | Address | # of filed Patents | Total Citations |
|---|---|---|---|
| Kaji, Akira | 1-9, Daimoncho 1-chome, Higashikurume-shi, Tokyo, 203, JP | 14 | 514 |
Cited Art
| Patent Info | (Count) | # Cites | Year |
|---|---|---|---|
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| 4,433,140 Tridecadeoxynucleotide, process for preparation thereof, and use thereof | 3 | 1982 | |
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| 4,464,359 (2'-5')-Oligo (3'-deoxyadenylate) and derivatives thereof | 19 | 1981 | |
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| 4,511,713 Process for selectively controlling unwanted expression or function of foreign nucleic acids in animal or mammalian cells | 89 | 1982 | |
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| 4,393,201 DNA Which codes for glycoprotein of era-strain rabies virus | 15 | 1981 | |
Patent Citation Ranking
Forward Cites
| Patent Info | (Count) | # Cites | Year |
|---|---|---|---|
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| 6,310,044 Oligonucleotide therapies for modulating the effects of herpesviruses | 5 | 1992 | |
| 5,580,767 Inhibition of influenza viruses by antisense oligonucleotides | 60 | 1992 | |
| 5,514,577 Oligonucleotide therapies for modulating the effects of herpes viruses | 63 | 1993 | |
| 5,639,595 Identification of novel drugs and reagents | 11 | 1993 | |
| 7,037,646 Amine-derivatized nucleosides and oligonucleosides | 3 | 1994 | |
| 5,643,780 Compositions and methods for modulating RNA activity through modification of the 5' cap structure of RNA | 5 | 1994 | |
| 5,658,891 Oligonucleotide therapies for modulating the effects of herpesviruses | 25 | 1994 | |
| 5,837,449 Compositions and methods for modulating .beta.-amyloid | 9 | 1994 | |
| 6,262,241 Compound for detecting and modulating RNA activity and gene expression | 17 | 1995 | |
| 5,852,182 Thiol-derivatized oligonucleosides | 12 | 1995 | |
| 5,872,232 2'-O-modified oligonucleotides | 41 | 1995 | |
| 5,859,221 2'-modified oligonucleotides | 70 | 1995 | |
| 5,587,469 Oligonucleotides containing N-2 substituted purines | 118 | 1995 | |
| 5,856,099 Antisense compositions and methods for modulating type I interleukin-1 receptor expression | 5 | 1996 | |
| 5,808,027 N-2 substituted purines in oligonucleotides | 2 | 1996 | |
| 6,077,833 Oligonucleotide compositions and methods for the modulation of the expression of B7 protein | 16 | 1996 | |
| 5,767,102 Antisense composition and method for treatment of CMV infection | 4 | 1997 | |
| 6,339,066 Antisense oligonucleotides which have phosphorothioate linkages of high chiral purity and which modulate .beta.I, .beta.II, .gamma., .delta., .EPSILON., .zeta. and .eta. isoforms of human protein kinase C | 0 | 1997 | |
| 5,985,558 Antisense oligonucleotide compositions and methods for the inibition of c-Jun and c-Fos | 29 | 1997 | |
| 5,965,722 Antisense inhibition of ras gene with chimeric and alternating oligonucleotides | 12 | 1997 | |
| 5,877,309 Antisense oligonucleotides against JNK | 51 | 1997 | |
| 6,001,991 Antisense oligonucleotide modulation of MDR P-glycoprotein gene expression | 3 | 1997 | |
| 6,005,087 2'-modified oligonucleotides | 56 | 1998 | |
| 6,528,631 Oligonucleotide-folate conjugates | 20 | 1998 | |
| 6,887,906 Compositions and methods for the delivery of oligonucleotides via the alimentary canal | 28 | 1998 | |
| 6,277,967 Carbohydrate or 2'-modified oligonucleotides having alternating internucleoside linkages | 12 | 1998 | |
| 6,242,589 Phosphorothioate oligonucleotides having modified internucleoside linkages | 16 | 1998 | |
| 6,232,463 Substituted purines and oligonucleotide cross-linking | 4 | 1998 | |
| 6,166,199 N-2 substituted purines | 0 | 1998 | |
| 6,221,850 Antisense oligonucleotide compositions and methods for the modulation of JNK proteins | 4 | 1998 | |
| 6,399,754 Sugar modified oligonucleotides | 10 | 1998 | |
| 6,177,246 Compositions and methods for modulating .beta.-amyloid | 7 | 1998 | |
| 6,359,124 Antisense inhibition of ras gene with chimeric and alternating oligonucleotides | 11 | 1999 | |
| 6,335,434 Nucleosidic and non-nucleosidic folate conjugates | 43 | 1999 | |
| 6,133,246 Antisense oligonucleotide compositions and methods for the modulation of JNK proteins | 60 | 1999 | |
| 6,369,209 Oligonucleotides having A-DNA form and B-DNA form conformational geometry | 10 | 1999 | |
| 8,153,602 Composition and methods for the pulmonary delivery of nucleic acids | 0 | 1999 | |
| 6,841,539 Compositions and methods for topical delivery of oligonucleotides | 11 | 1999 | |
| 6,319,906 Oligonucleotide compositions and methods for the modulation of the expression of B7 protein | 10 | 1999 | |
| 6,656,730 Oligonucleotides conjugated to protein-binding drugs | 18 | 1999 | |
| 6,326,358 Carbohydrate or 2'-modified oligonucleotides having alternating internucleoside linkages | 14 | 1999 | |
| 6,440,943 Oligonucleotides having site specific chiral phosphorothioate internucleoside linkages | 11 | 1999 | |
| 6,312,900 Antisense oligonucleotide compositions and methods for the modulation of activating protein 1 | 3 | 1999 | |
| 6,265,558 Thiol-derivatized nucleosides and oligonucleosides | 10 | 1999 | |
| 6,531,584 2'modified oligonucleotides | 42 | 1999 | |
| 6,653,458 Modified oligonucleotides | 7 | 1999 | |
| 6,867,294 Gapped oligomers having site specific chiral phosphorothioate internucleoside linkages | 3 | 1999 | |
| 6,753,423 Compositions and methods for enhanced biostability and altered biodistribution of oligonucleotides in mammals | 3 | 2000 | |
| 6,762,169 Ligand-conjugated oligomeric compounds | 6 | 2000 | |
| 6,809,193 Antisense oligonucleotide compositions and methods for the modulation of JNK proteins | 14 | 2001 | |
| 6,811,975 Phosphorothioate oligonucleotides having modified internucleoside linkages | 6 | 2001 | |
| 7,056,896 Carbohydrate or 2'-modified oligonucleotides having alternating internucleoside linkages | 1 | 2001 | |
| 7,119,184 Oligonucleotides having A-DNA form and B-DNA form conformational geometry | 0 | 2001 | |
| 6,861,514 Nucleosidic and non-nucleosidic folate conjugates | 2 | 2001 | |
| 7,138,517 Sugar modified oligonucleotides | 8 | 2001 | |
| 6,537,973 Oligonucleotide inhibition of protein kinase C | 5 | 2001 | |
| 6,747,014 Compositions and methods for non-parenteral delivery of oligonucleotides | 20 | 2001 | |
| 7,695,902 Oligoribonucleotides and ribonucleases for cleaving RNA | 3 | 2002 | |
| 6,737,520 Oligonucleotides having A-DNA form and B-DNA form conformational geometry | 0 | 2002 | |
| 6,919,439 Derivatized oligonucleotides having improved uptake and other properties | 0 | 2002 | |
| 7,235,650 Derivatized oligonucleotides having improved uptake and other properties | 0 | 2002 | |
| 7,235,653 Oligonucleotide compositions and methods for the modulation of the expression of B7 protein | 2 | 2003 | |
| 7,812,149 2′-Fluoro substituted oligomeric compounds and compositions for use in gene modulations | 0 | 2003 | |
| 8,084,432 Compositions and methods for treatment of pouchitis | 0 | 2004 | |
| 8,394,947 Positionally modified siRNA constructs | 0 | 2004 | |
| 7,960,355 Compositions and methods for the modulation of the expression of B7 protein | 0 | 2004 | |
| RE39464 Oligonucleolotides having site specific chiral phosphorothioate internucleoside linkages | 2 | 2004 | |
| 7,884,086 Conjugates for use in hepatocyte free uptake assays | 1 | 2005 | |
| 8,377,897 Compositions and methods for non-parenteral delivery of oligonucleotides | 0 | 2005 | |
| 7,897,582 Oligonucleotide compositions and methods for the modulation of the expression of B7 protein | 0 | 2007 | |
| 8,101,585 Compositions and methods for the modulation of JNK proteins | 0 | 2007 | |
| 7,964,579 Compositions and methods for topical delivery of oligonucleotides | 0 | 2009 | |
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| 5,703,055 Generation of antibodies through lipid mediated DNA delivery | 173 | 1994 | |
| 5,580,859 Delivery of exogenous DNA sequences in a mammal | 460 | 1994 | |
| 5,589,466 Induction of a protective immune response in a mammal by injecting a DNA sequence | 340 | 1995 | |
| 6,673,776 Expression of exogenous polynucleotide sequences in a vertebrate, mammal, fish, bird or human | 1 | 1995 | |
| 5,693,622 Expression of exogenous polynucleotide sequences cardiac muscle of a mammal | 138 | 1995 | |
| 6,228,844 Stimulating vascular growth by administration of DNA sequences encoding VEGF | 18 | 1997 | |
| 6,710,035 Generation of an immune response to a pathogen | 10 | 1999 | |
| 6,413,942 Methods of delivering a physiologically active polypeptide to a mammal | 38 | 1999 | |
| 6,706,694 Expression of exogenous polynucleotide sequences in a vertebrate | 9 | 2000 | |
| 7,250,404 Lipid-mediated polynucleotide administration to deliver a biologically active peptide and to induce a cellular immune response | 9 | 2002 | |
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| 8,067,383 Synthetic genes and genetic constructs comprising same I | 2 | 2003 | |
| 7,754,697 Control of gene expression | 10 | 2003 | |
| 8,048,670 Synthetic genes and genetic constructs | 4 | 2004 | |
| 7,855,071 Synthetic genes and genetic constructs | 0 | 2004 | |
| 8,053,419 Synthetic genes and genetic constructs | 4 | 2004 | |
| 8,183,217 Methods and means for obtaining modified phenotypes | 5 | 2005 | |
| 8,168,774 Control of gene expression | 4 | 2005 | |
| 8,431,547 Synthetic genes and genetic constructs | 0 | 2011 | |
| 8,334,374 Methods and means for obtaining modified phenotypes | 0 | 2012 | |
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| 5,733,781 Oligonucleotides and methods for inhibiting propagation of human immunodeficiency virus | 2 | 1994 | |
| 5,629,413 Oligonucleotides with activity against human immunodeficiency virus | 13 | 1994 | |
| 5,739,309 Enhancement of oligonucleotide inhibition of protein production, cell proliferation and / or multiplication of infectious disease pathogens | 20 | 1995 | |
| 5,919,701 Oligonucleotides with activity against human immunodeficiency virus | 13 | 1997 | |
| 5,874,281 Enhancement of oligonucleotide inhibition of protein production, cell proliferation, and/or multiplication of infectious disease pathogens | 2 | 1997 | |
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| 5,739,308 Integrated oligonucleotides | 11 | 1995 | |
| 5,929,226 Antisense oligonucleotide alkylphosphonothioates and arylphospohonothioates | 27 | 1995 | |
| 5,750,674 Methods and compounds for the stereoselective enrichment of oligonucleotide diastereomers and oligonucleotides thereby produced | 2 | 1995 | |
| 5,693,773 Triplex-forming antisense oligonucleotides having abasic linkers targeting nucleic acids comprising mixed sequences of purines and pyrimidines | 35 | 1995 | |
| 6,117,993 Synthons for oligonucleotide synthesis | 2 | 1998 | |
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| 7,335,765 Nucleoside and oligonucleotide analogues | 5 | 2001 | |
| 7,217,805 Bicyclonucleoside analogues | 10 | 2002 | |
| 7,314,923 Nucleoside and oligonucleotide analogues | 10 | 2003 | |
| 7,816,333 Oligonucleotide analogues and methods utilizing the same | 1 | 2007 | |
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| 5,637,573 Influenza virus replication inhibiting oligonucleotide analogues and their pharmaceutical compositions | 9 | 1995 | |
| 6,683,167 Hybrid oligonucleotide phosphorothioates | 18 | 2001 | |
| 7,045,609 Hybrid oligonucleotide phosphorothioates | 15 | 2002 | |
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| 5,610,050 Methods of preventing viral replication | 2 | 1993 | |
| 6,001,990 Antisense inhibition of hepatitis C virus | 13 | 1995 | |
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| 5,177,198 Process for preparing oligoribonucleoside and oligodeoxyribonucleoside boranophosphates | 58 | 1989 | |
| 5,455,233 Oligoribonucleoside and oligodeoxyribonucleoside boranophosphates | 113 | 1992 | |
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| 6,867,195 Lipid-mediated polynucleotide administration to reduce likelihood of subject's becoming infected | 9 | 1995 | |
| 6,214,804 Induction of a protective immune response in a mammal by injecting a DNA sequence | 154 | 1995 | |
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| 4,806,463 Inhibition of HTLV-III by exogenous oligonucleotides | 211 | 1986 | |
| 5,194,428 Inhibition of influenza virus replication by oligonucleotide phosphorothioates | 130 | 1990 | |
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| 5,837,852 Capped nucleic acid oligomers that inhibit cap-dependent transcription of the influenza virus endonuclease | 5 | 1993 | |
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| 7,449,449 Particle-mediated transformation of vertebrate tissue cells | 0 | 2003 | |
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| 7,358,234 Induction of a protective immune response through microprojectiles coated with a DNA sequence encoding an immunogenic protein | 0 | 2003 | |
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| 6,015,676 Method for knocking out gene transcripts by covalently binding of an anti-sense probe | 5 | 1998 | |
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| 6,033,909 Oligonucleotide analogs, their preparation and use | 16 | 1994 | |
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| 6,346,614 Hybrid oligonucleotide phosphorothioates | 45 | 2000 | |
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| 6,995,008 Coordinate in vivo gene expression | 1 | 1999 | |
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| 5,474,935 Adeno-associated virus (AAV)-based eucaryotic vectors | 91 | 1993 | |
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| 5,135,917 Interleukin receptor expression inhibiting antisense oligonucleotides | 96 | 1990 | |
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| 6,306,831 Transplacental delivery of oligonucleotides | 1 | 1998 | |
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| 6,576,218 Transplacental delivery of oligonucleotides | 0 | 2001 | |
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| 5,004,810 Antiviral oligomers | 100 | 1988 | |
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| 4,904,582 Novel amphiphilic nucleic acid conjugates | 135 | 1987 | |
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| 7,994,145 Bicyclonucleoside analogues | 0 | 2007 | |
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| 5,098,890 Antisence oligonucleotides to c-myb proto-oncogene and uses thereof | 133 | 1989 | |
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| 5,942,389 Genes and genetic elements associated with sensitivity to cisplatin | 3 | 1995 | |
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| 5,834,185 Formation of triple helix complexes of single stranded nucleic acids using nucleoside oligomers which comprise pyrimidine analogs, triple helix complexes formed thereby and oligomers used in their formation | 12 | 1994 | |
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| 7,704,965 Methods and materials for treating human papillomavirus infections | 0 | 2003 | |
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| 6,806,084 Methods for compositions for in vivo gene delivery | 0 | 1998 | |
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| 6,521,601 Method and composition for inhibition of viral replication | 2 | 1992 | |
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| 6,143,881 Hybrid oligonucleotide phosphorothioates | 42 | 1995 | |
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| 5,885,834 Antisense oligodeoxynucleotide against phosphodiesterase | 13 | 1997 | |
Maintenance Fees
| Fee | Large entity fee | small entity fee | micro entity fee | due date |
|---|
| Fee | Large entity fee | small entity fee | micro entity fee |
|---|---|---|---|
| Surcharge after expiration - Late payment is unavoidable | $700.00 | $350.00 | $175.00 |
| Surcharge after expiration - Late payment is unintentional | $1,640.00 | $820.00 | $410.00 |