US Patent No: 7,417,022

Number of patents in Portfolio can not be more than 2000

Compounds and compositions for delivering active agents

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ALSO PUBLISHED AS: 20050186176
ATTORNEY / AGENT: (SPONSORED)
 

Importance

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Abstract

Modified amino acid compounds useful in the delivery of active agents are provided. Methods of administration and preparation are provided as well.

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First Claim

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Patent Owner(s)

Patent OwnerAddressTotal Patents
MHR INSTITUTIONAL PARTNERS IIA LPNEW YORK, NY2

International Classification(s)

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  • [Patents Count]

Inventor(s)

Inventor Name Address # of filed Patents Total Citations
Leipold, Harry Elmsford, NY 19 445
Leone-Bay, Andrea Ridgefield, CT 120 1978
Milstein, Sam J Larchmont, NY 60 1535
Sarubbi, Donald J Bolton, MA 53 1146

Cited Art

Patent Info (Count) # Cites Year
 
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4,925,673 Delivery systems for pharmacological agents encapsulated with proteinoids 259 1987
4,895,725 Microencapsulation of fish oil 97 1988
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4,983,402 Orally administerable ANF 79 1989
5,443,841 Proteinoid microspheres and methods for preparation and use thereof 62 1992
5,401,516 Modified hydrolyzed vegetable protein microspheres and methods for preparation and use thereof 55 1993
5,451,410 Modified amino acids for encapsulating active agents 88 1993
5,578,323 Proteinoid carriers and methods for preparation and use thereof 77 1993
5,447,728 Desferrioxamine oral delivery system 75 1993
5,792,451 Oral drug delivery compositions and methods 85 1994
5,541,155 Acids and acid salts and their use in delivery systems 91 1994
5,629,020 Modified amino acids for drug delivery 95 1994
5,540,939 Modified hydrolyzed vegetable protein microspheres and methods for preparation and use thereof 48 1994
5,643,957 Compounds and compositions for delivering active agents 89 1994
5,714,167 Active agent transport systems 62 1994
5,972,387 Modified hydrolyzed vegetable protein microspheres and methods for preparation and use thereof 17 1994
5,709,861 Compositions for the delivery of antigens 62 1995
5,650,386 Compositions for oral delivery of active agents 85 1995
5,820,881 Microspheres of diamide-dicarboxylic acids 31 1995
5,601,846 Proteinoid microspheres and methods for preparation and use thereof 66 1995
5,958,457 Compositions for the delivery of antigens 38 1995
6,180,140 Modified amino acids for drug delivery 29 1995
5,667,806 Spray drying method and apparatus 66 1995
5,750,147 Method of solubilizing and encapsulating itraconazole 58 1995
5,824,345 Fragrances and flavorants 27 1995
6,051,258 Proteinoid emulsions and methods for preparation and use thereof 32 1995
5,811,127 Desferrioxamine oral delivery system 54 1996
5,840,340 Proteinoid carriers and methods for preparation and use thereof 26 1996
5,935,601 Modified amino acids for drug delivery 31 1996
6,099,856 Active agent transport systems 42 1996
5,866,536 Compounds and compositions for delivering active agents 54 1997
5,955,503 Compounds and compositions for delivering active agents 26 1997
5,965,121 Compounds and compositions for delivering active agents 34 1997
5,989,539 Compounds and compositions for delivering active agents 32 1997
6,001,347 Compounds and compositions for delivering active agents 42 1997
6,100,298 Compounds and compositions for delivering active agents 31 1997
5,773,647 Compounds and compositions for delivering active agents 61 1997
5,776,888 Compounds and compositions for delivering active agents 43 1997
5,804,688 Compounds and compositions for delivering active agents 33 1997
5,876,710 Compounds and compositions for delivering active agents 34 1997
5,879,681 Compounds and compositions for delivering active agents 35 1997
5,939,381 Compounds and compositions for delivering active agents 27 1997
5,990,166 Compounds and compositions for delivering active agents 37 1997
6,051,561 Compounds and compositions for delivering active agents 35 1997
6,060,513 Compounds and compositions for delivering active agents 36 1997
6,090,958 Compounds and compositions for delivering active agents 36 1997
6,358,504 Compounds and compositions for delivering active agents 18 1997
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6,348,207 Orally deliverable supramolecular complex 17 1997
6,100,285 Method of solubilizing itraconazole 25 1997
6,084,112 Method for preparing .omega.-aminoalkanoic acid derivatives from cycloalkanones 19 1997
6,391,303 Methods and compositions for inducing oral tolerance in mammals 11 1999
6,428,780 Compounds and compositions for delivering active agents 14 1999
6,346,242 Compounds and compositions for delivering active agents 21 2000
6,384,278 Boron-mediated amidation of carboxylic acids 11 2001
6,642,411 Compounds and compositions for delivering active agents 13 2001
6,440,929 Pulmonary delivery of active agents 13 2001
6,461,643 Oral drug delivery compositions and methods 17 2001
6,610,329 Compositions for the delivery of antigens 15 2001
6,399,798 Method of preparing alkylated salicylamides 18 2001
6,646,162 Compounds and compositions for delivering active agents 14 2001
6,623,731 Compounds and compositions for delivering active agents 12 2001
6,525,020 Compounds and compositions for delivering active agents 12 2001
6,663,887 Compounds and compositions for delivering active agents 11 2002
6,699,467 Compounds and compositions for delivering active agents 14 2002
6,693,073 Pulmonary delivery of active agents 12 2002
6,693,208 Compounds and compositions for delivering active agents 14 2002
2005/0272,815 Compounds and compositions for delivering active agents 1 2005
 
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CONNAUGHT LABORATORIES LIMITED (2)
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4,837,381 Compositions for parenteral administration and their use 76 1987
 
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BAHN, PETER, FARMINGTON, CT, (5.0%) INTEREST (1)
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Bayer Aktiengesellschaft (1)
4,402,856 Microcapsules with a defined opening temperature, a process for their production and their use 109 1981
 
Biomaterials Universe, Inc. (1)
5,100,669 Polylactic acid type microspheres containing physiologically active substance and process for preparing the same 169 1989
 
BIOTECHNOLOGY MANAGEMENT ASSOCIATES, INCORPORATED (1)
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Blue Wing Corporation (1)
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BOEHRINGER BIOCHEMIA ROBIN S.P.A. (1)
4,753,804 Granular dietetic product based on amino acids and process for their preparation 75 1985
 
Boehringer Mannheim GmbH (1)
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Ceskoslovenska akademie ved (1)
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Choay S.A. (1)
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CIBA-GEIGY CORPORATION (1)
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Clean Air, Inc. (1)
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CLEAR LAKE DEVELOPMENT GROUP, 201 N. MAIN, WICHITA, KN., 67202 A PARTNERSHIP (1)
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COLLAGEN MATRIX TECHNOLOGIES, INC. (1)
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CRYOGENIC TECHNOLOGY, INC. (1)
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DAINIPPON PHARMACEUTICAL CO., LTD. (1)
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Dr. Wolman GmbH (1)
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EURAND S.P.A. (1)
4,460,563 Process for preparing microcapsules in a liquid vehicle 85 1981
 
Farmaceutici Formenti S.p.A. (1)
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Fisons Limited (1)
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5,216,124 Substituted cyclic tetrapeptides 59 1991
 
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INNOVATA BIOMED LIMITED (1)
5,384,133 Pharmaceutical formulations comprising microcapsules 161 1993
 
INTERx Research Corporation (1)
4,462,991 Method of increasing oral absorption of polar bioactive agents 87 1982
 
ISP Chemicals Inc. (1)
5,244,653 Glycine anhydride dimethylol as a biocide and preservative 61 1991
 
Japan Atomic Energy Research Institute (1)
4,483,807 Process for producing a slow release composite 75 1982
 
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Kyoto Yakuhin Kogyo Kabushiki Kaisha (1)
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La Jolla Cancer Research Foundation (1)
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Lion Corporation (1)
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5,705,529 N-benzoyl amino acid derivatives pharmaceutical compositions containing them and process for preparing same 68 1995
 
Nitto Electric Industrial Co., Ltd. (1)
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Nordisk Insulinlaboratorium (1)
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PHARMETRIX, MENLO PARK (1)
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4,647,455 Process for extracting atrial natriuretic factor 63 1984
 
REAADS MEDICAL PRODUCTS, INC., A DE CORP. (1)
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REVLON CONSUMER PRODUCTS CORPORATION (1)
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Rhone-Poulenc Chimie (1)
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SANKYO COMPANY, LIMITED (1)
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Other [Check patent profile for assignment information] (4)
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4,708,952 Method of treatment of the infectious and viral diseases by one time interference 57 1986
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