Pharmaceutical salts of macrocyclic modulators of the ghrelin receptor

Number of patents in Portfolio can not be more than 2000

United States of America Patent

PATENT NO 8334256
APP PUB NO 20090221689A1
SERIAL NO

12351395

Stats

ATTORNEY / AGENT: (SPONSORED)

Importance

Loading Importance Indicators... loading....

Abstract

See full text

The present invention provides novel conformationally-defined macrocyclic compounds that have been demonstrated to be selective modulators of the ghrelin receptor (growth hormone secretagogue receptor, GHS-R1a and subtypes, isoforms and variants thereof). Methods of synthesizing the novel compounds are also described herein. These compounds are useful as agonists of the ghrelin receptor and as medicaments for treatment and prevention of a range of medical conditions including, but not limited to, metabolic and/or endocrine disorders, gastrointestinal disorders, cardiovascular disorders, obesity and obesity-associated disorders, central nervous system disorders, genetic disorders, hyperproliferative disorders and inflammatory disorders.

Loading the Abstract Image... loading....

First Claim

See full text

Family

Loading Family data... loading....

Patent Owner(s)

Patent OwnerAddress
OCERA THERAPEUTICS INC525 UNIVERSITY AVENUE STE 610 PALO ALTO CA 94301-1920

International Classification(s)

Inventor(s)

Inventor Name Address # of filed Patents Total Citations
Marsault, Eric Québec, CA 40 487
St-Louis, Carl Québec, CA 9 74

Cited Art Landscape

Load Citation

Patent Citation Ranking

Forward Cite Landscape

Load Citation