Kappa opioid receptor agonists

Number of patents in Portfolio can not be more than 2000

United States of America Patent

PATENT NO 9303027
APP PUB NO 20130303525A1
SERIAL NO

13811020

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Abstract

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The present invention relates to a series of substituted compounds having the general formula (I), including their stereoisomers and/or their pharmaceutically acceptable salts. (I) Wherein A, m, R1s, R2, R3, R4 are as defined herein. This invention also relates to methods of making these compounds including intermediates. The compounds of this invention are effective at the kappa (κ) opioid receptor (KOR) site. Therefore, the compounds of this invention are useful as pharmaceutical agents, especially in the treatment and/or prevention of a variety of central nervous system disorders (CNS), including but not limited to acute and chronic pain, and associated disorders, particularly functioning peripherally at the CNS.

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Patent Owner(s)

Patent OwnerAddress
DR REDDY'S LABORATORIES INC200 SOMERSET CORPORATE BLVD 7TH FLOOR BRIDGEWATER NJ 08807
DR REDDY'S LABORATORIES LTDHYDERABAD 500 034

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Inventor(s)

Inventor Name Address # of filed Patents Total Citations
Chintakunta, Vamsee Krishna Hyderabad, IN 3 6
Elster, Lisbeth Herlev, DK 1 1
Frimurer, Thomas Michael Copenhagen S., DK 2 4
Gerlach, Lars-Ole Vedbaek, DK 4 10
Hogberg, Thomas Akarp, SE 17 128
Jaleel, Mahaboobi Hyderabad, IN 1 1
Khanna, Ish Kumar Alpharetta, US 26 178
Potluri, Vijay Hyderabad, IN 16 35
Rist, Oystein Ballerup, DK 5 56
Sasmal, Pradip Kumar Hyderabad, IN 15 57
Tehim, Ashok Ridgewood, US 111 824

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