C-3 ALKYL AND ALKENYL MODIFIED BETULINIC ACID DERIVATIVES USEFUL IN THE TREATMENT OF HIV

European Patent Office Patent

APP PUB NO EP-2958930-A1
SERIAL NO

14710687

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Abstract

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Compounds having drug and bio-affecting properties, their pharmaceutical compositions and methods of use are set forth. In particular, alkyl and alkenyl C-3 modified betulinic acid derivatives that possess unique antiviral activity are provided as HIV maturation inhibitors, as represented by compounds of Formulas I, II, III and IV: a compound of Formula I; a compound of Formula II; a compound of Formula III: and a compound of Formula IV. These compounds are useful for the treatment of HIV and AIDS.

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Patent Owner(s)

Patent OwnerAddress
BRISTOL MYERS SQUIBB COUSROUTE 206 AND PROVINCE LINE ROAD PRINCETON NEW JERSEY 08543 US

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Inventor(s)

Inventor Name Address
MEANWELL NICHOLAS A EAST HAMPTON CT 06424
REGUEIRO-REN ALICIA C/O BRISTOL-MYERS SQUIBB COMPANY ROUTE 206 AND PROVINCE LINE ROAD PRINCETON NEW JERSEY 08543 US
SWIDORSKI JACOB WALLINGFORD CONNECTICUT 06492
HARTZ RICHARD A KENNETT SQUARE PA 19348
CHEN YAN SEATTLE WA 98109
XU LI SPRINGFIELD ILLINOIS 62711
LIU ZHENG INGLEWOOD CALIFORNIA 90301
SIT SING-YUEN MERIDEN CT 06450
CHEN JIE SNELLVILLE GEORGIA 30078

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