LACTAM-CONTAINING COMPOUNDS AND DERIVATIVES THEREOF AS FACTOR XA INHIBITORS

World Intellectual Property Organization Patent

APP PUB NO WO-2003026652-A1
SERIAL NO

PCTUS0229491

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Abstract

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The present application describes lactam-containing compounds and derivatives thereof of Formula I: P4-P-M-M4 or pharmaceutically acceptable salt forms thereof, wherein ring P, if present is a 5-7 membered carbocycle or heterocycle and ring M is a 5-7 membered carbocycle or heterocycle. Compounds of the present invention are useful as inhibitors of trypsin-like serine proteases, specifically factor Xa.

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Patent Owner(s)

Patent OwnerAddress
BRISTOL MYERS SQUIBB COUSP O BOX 4000 ROUTE 206 AND PROVINCE LINE ROAD PRINCETON NJ 08543-4000 US

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Inventor(s)

Inventor Name Address
LI YUN-LONG WILMINGTON DELAWARE 19803
HAN WEI 17021 ALDINE WESTFIELD ROAD HOUSTON TEXAS 77073 77073
PINTO DONALD 425 BRENTFORD ROAD KENNETT SQUARE PA 19348
QIAO JENNIFER 22D PRESIDENTIAL DRIVE WILMINGTON DE 19807
ORWAT MICHAEL 18 S COLTS NECK WAY HOCKESSIN DE 19707
QUAN MIMI 113 VENUS DRIVE NEWARK DE 19711
LAM PATRICK 6 RIDGEWAY DRIVE CHADDS FORD PA 19317
KOCH STEPHANIE 7 FEDERAL FARM DRIVE BOOTHWYN PA 19061

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