LACTAM-CONTAINING COMPOUNDS AND DERIVATIVES THEREOF AS FACTOR XA INHIBITORS

World Intellectual Property Organization Patent

APP PUB NO WO-2003026652-A1
SERIAL NO

PCTUS0229491

Stats

Importance

Loading Importance Indicators... loading....

Abstract

See full text

The present application describes lactam-containing compounds and derivatives thereof of Formula I: P4-P-M-M4 or pharmaceutically acceptable salt forms thereof, wherein ring P, if present is a 5-7 membered carbocycle or heterocycle and ring M is a 5-7 membered carbocycle or heterocycle. Compounds of the present invention are useful as inhibitors of trypsin-like serine proteases, specifically factor Xa.

Loading the Abstract Image... loading....

First Claim

See full text

Family

Loading Family data... loading....

Patent Owner(s)

Patent OwnerAddress
BRISTOL MYERS SQUIBB COUSRTE 206 & PROVINCE LINE ROAD PRINCETON NEW JERSEY 08543 US

International Classification(s)

Inventor(s)

Inventor Name Address
LI YUN-LONG CHADDS FORD PA
HAN WEI PORTLAND OR
PINTO DONALD KENNETT SQUARE PA 19348
QIAO JENNIFER PRINCETON NJ
ORWAT MICHAEL NEW HOPE PA 18938
QUAN MIMI YARDLEY PA 19067
LAM PATRICK CHADDS FORD PA 19317
KOCH STEPHANIE NEWARK DE 19711

Cited Art Landscape

Load Citation