MONOCLONAL ANTIBODIES AGAISNT ACTIVATED PROTEIN C (aPC)

World Intellectual Property Organization Patent

APP PUB NO WO-2014085596-A1
SERIAL NO

PCTWO2013072243

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Abstract

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Provided herein are antibodies, antigen-binding antibody fragments (Fabs), and other protein scaffolds, directed against human activated Protein C (aPC) with minimal binding to its zymogen Protein C (PC). Moreover, these aPC binding proteins could potentially block the anti-coagulant activity of aPC to induce coagulation. Therapeutic uses of these binders are described herein as are methods of panning and screening specific antibodies.

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Patent Owner(s)

Patent OwnerAddress
BAYER HEALTHCARE LLCUSNEW JERSEY NEW JERSEY

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Inventor(s)

Inventor Name Address
WILMEN ANDREAS ARNDTSTR 5 50676 KÖLN
MURPHY JOHN E BERKELEY CALIFORNIA 94707
WANG ZHUOZHI MILLBRAE CALIFORNIA 94030
GU JIAN-MING LAFAYETTE CA
MCLEAN KIRK FULLERTON CA
BAUZON MAXINE HERCULES CALIFORNIA 94547
MARQUARDT TOBIAS WUPPERTAL
KIM JI-YUN BERKELEY CA
ZHAO XIAO-YAN UNION CITY CA
JIN FANG C/O PFIZER INC 610 MAIN STREET CAMBRIDGE MASSACHUSETTS 02139 02139
WANG XINQUAN 310003 THREE UNITS 1901 WANDA COMMERCIAL CENTER GONGSHU DISTRICT HANGZHOU CITY ZHEJIANG PROVINCE HANGZHOU CITY ZHEJIANG PROVINCE 310003

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