SPIRO COMPOUNDS AS MELANOCORTIN 4 RECEPTOR ANTAGONISTS AND USES THEREOF

World Intellectual Property Organization Patent

APP PUB NO WO-2021250541-A1
SERIAL NO

PCTIB2021054970

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Abstract

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Described herein are compounds of Formula I and their pharmaceutically acceptable salts, wherein R1, R2, R3, X1, Y1, Y2, Y3, Y4 and Y5 are defined herein; their use as MC4R antagonists; pharmaceutical compositions containing such compounds and salts; the use of such compounds and salts to treat, for example, cachexia, anorexia, or anorexia nervosa; and intermediates and processes for preparing such compounds and salts.

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Patent Owner(s)

Patent OwnerAddress
PFIZERUS235 EAST 42ND STREET NEW YORK NY 10017 US

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Inventor(s)

Inventor Name Address
BUTLER CHRISTOPHER RYAN CANTON MA 02021
SMITH AARON CHRISTOPHER MARIETTA GA
POLIVKOVA JANA MYSTIC CT
SAMMONS MATTHEW FORREST QUINCY MA
GARNSEY MICHELLE RENEE PROVIDENCE RHODE ISLAND 02906
YANG QINGYI LEXINGTON MA 02420
OGILVIE KEVIN ALEXANDER GALES FERRY CT

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