C07D 203/04

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Patent/Pub #TitleFiling DateIssue/Publication DatePatent Owner
2024/0408,215 USE OF DIAZIRINE LINKER FOR DRUG CONJUGATESSep 08, 22Dec 12, 24Helmholtz Zentrum Munchen Deutsches Forschungszentrum fur Gesundheit und Umwelt (GmbH)
2024/0397,813 ORGANIC COMPOUND, AND ORGANIC LIGHT-EMITTING DEVICE COMPRISING SAMESep 27, 21Nov 28, 24P&H TECH Co., Ltd
2024/0092,742 REAGENT FOR MASS SPECTROMETRYNov 02, 23Mar 21, 24Not available
2024/0067,600 SMALL MOLECULE INHIBITORS OF THE MITOCHONDRIAL PERMEABILITY TRANSITION PORE (mtPTP)Mar 16, 23Feb 29, 24The University of Kansas; Oregon Health & Science University;
2023/0234,920 Azirine Containing Compounds as Anti-Angiogenesis Agents and a Process for the Preparation ThereofJun 04, 21Jul 27, 23Not available
2022/0089,537 HIGH-THROUGHPUT METHOD TO RAPIDLY ADD CHEMICAL MOIETIES TO A SMALL MOLECULE LIBRARYJul 12, 21Mar 24, 22Massachusetts Institute of Technology; President and Fellows of Harvard College;
2018/0282,264 SMALL MOLECULE INHIBITORS OF THE MITOCHONDRIAL PERMEABILITY TRANSITION PORE (mtPTP)Nov 04, 15Oct 04, 18Not available
2012/0208,918 STABILIZATION OF COMPOUNDS COMPRISING IODINEMar 25, 10Aug 16, 12LANXESS DEUTSCHLAND GMBH
2011/0112,254 POLYMERIC COMPOSITIONS AND METHOD OF MAKING AND ARTICLES THEREOFNov 10, 10May 12, 113M INNOVATIVE PROPERTIES COMPANY
2010/0273,762 Method of combating infectionSep 04, 06Oct 28, 10MORVUS TECHNOLOGY LIMITED
2010/0215,574 PROCESS FOR PRODUCING AN INJECTABLE MEDICAMENT PREPARATIONOct 22, 09Aug 26, 10KTB TUMORFORSCHUNGS GMBH
2010/0081,759 ACRYLIC PRESSURE-SENSITIVE ADHESIVES WITH AZIRIDINE CROSSLINKING AGENTSDec 08, 09Apr 01, 103M INNOVATIVE PROPERTIES COMPANY
2010/0056,806 C-H Bond Amination and Olefin Aziridination with Beta-Diketiminato Copper CatalystsDec 05, 07Mar 04, 10GEORGETOWN UNIVERSITY
2009/0208,740 ACRYLIC PRESSURE-SENSITIVE ADHESIVES WITH AZIRIDINE CROSSLINKING AGENTSFeb 14, 08Aug 20, 093M INNOVATIVE PROPERTIES COMPANY
2007/0232,581 Oxime-Containing Acyl Guanidines as Beta-Secretase InhibitorsMar 29, 07Oct 04, 07BRISTOL-MYERS SQUIBB COMPANY
2005/0222,081 Cross-linked hyaluronate compoundsMay 04, 05Oct 06, 05Not available
2004/0220,413 Method of producing optically active aziridine compounds and amine compoundsFeb 06, 04Nov 04, 04KYUSHU UNIVERSITY, NATIONAL UNIVERSITY CORPORATION
2003/0204,098 Method for production of aziridines and N-vinylamidesApr 10, 03Oct 30, 03NIPPON SHOKUBAI CO., LTD.
2003/0166,634 Unsaturated 1-Amino-alkylcyclohexane NMDA, 5HT3, and neuronal nicotinic receptor antagonistsNov 06, 02Sep 04, 03MERZ PHARMA GMBH & CO. KGAA
2003/0153,771 Large scale synthesis of optically pure aziridinesSep 27, 02Aug 14, 03LEXICON PHARMACEUTICALS, INC.

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